sotuletinib [Ligand Id: 8250] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| platelet derived growth factor receptor beta in Human [GtoPdb: 1804] [UniProtKB: P09619] | ||||||||
| GtoPdb | - | - | 5.23 | pIC50 | 5860 | nM | IC50 | Oncoimmunology (2013) 2: e26968 [PMID:24498562] |
| KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721] | ||||||||
| GtoPdb | - | - | 5.41 | pIC50 | 3880 | nM | IC50 | Oncoimmunology (2013) 2: e26968 [PMID:24498562] |
| colony stimulating factor 1 receptor in Human [GtoPdb: 1806] [UniProtKB: P07333] | ||||||||
| GtoPdb | - | - | 8.47 | pKd | 3.4 | nM | Kd | J Med Chem (2020) 63: 9888-9911 [PMID:32787110] |
| GtoPdb | - | - | 9 | pIC50 | 1 | nM | IC50 | Oncoimmunology (2013) 2: e26968 [PMID:24498562] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
