SGC-CBP30 [Ligand Id: 7529] activity data from GtoPdb

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  • CREB binding lysine acetyltransferase in Human [GtoPdb: 2734] [UniProtKB: Q92793]
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  • EP300 lysine acetyltransferase in Human [GtoPdb: 2735] [UniProtKB: Q09472]
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  • Plasmodium falciparum histone acetyltransferase GCN5 in Plasmodium falciparum Dd2 [GtoPdb: 3191]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CREB binding lysine acetyltransferase in Human [GtoPdb: 2734] [UniProtKB: Q92793]
GtoPdb - - 7.16 pIC50 69 nM IC50 ChemMedChem (2014) 9: 438-64 [PMID:24497428]
EP300 lysine acetyltransferase in Human [GtoPdb: 2735] [UniProtKB: Q09472]
GtoPdb - - 7.42 pIC50 38 nM IC50 ChemMedChem (2014) 9: 438-64 [PMID:24497428]
Plasmodium falciparum histone acetyltransferase GCN5 in Plasmodium falciparum Dd2 [GtoPdb: 3191]
GtoPdb Parasite growth inhibition assay - 5.5 pIC50 3160 nM IC50 Int J Parasitol Drugs Drug Resist (2018) 8: 189-193 [PMID:29631126]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.