SU-14813 [Ligand Id: 5712] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| platelet derived growth factor receptor beta in Human [GtoPdb: 1804] [UniProtKB: P09619] | ||||||||
| GtoPdb | - | - | 8.4 | pIC50 | 4 | nM | IC50 | Mol Cancer Ther (2006) 5: 1774-82 [PMID:16891463] |
| KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721] | ||||||||
| GtoPdb | - | - | 7.82 | pIC50 | 15 | nM | IC50 | Mol Cancer Ther (2006) 5: 1774-82 [PMID:16891463] |
| fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362] | ||||||||
| GtoPdb | - | - | 5.46 | pIC50 | 3500 | nM | IC50 | Mol Cancer Ther (2006) 5: 1774-82 [PMID:16891463] |
| fms related receptor tyrosine kinase 1 in Human [GtoPdb: 1812] [UniProtKB: P17948] | ||||||||
| GtoPdb | - | - | 8.7 | pIC50 | 2 | nM | IC50 | Mol Cancer Ther (2006) 5: 1774-82 [PMID:16891463] |
| kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968] | ||||||||
| GtoPdb | - | - | 8.64 | pKd | 2.3 | nM | Kd | Nat Biotechnol (2011) 29: 1046-51 [PMID:22037378] |
| GtoPdb | - | - | 7.3 | pIC50 | 50 | nM | IC50 | Mol Cancer Ther (2006) 5: 1774-82 [PMID:16891463] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
