capeserod [Ligand Id: 29] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL2027925 (Sl65.0155, SL650155, Capeserod)
  • 5-HT1A receptor in Human [GtoPdb: 1] [UniProtKB: P08908]
  • This target only has 1 pki data point
  • 6
1 CHEMBL2027925_lig_chart_1 5-HT1A receptor Human
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  • 5-HT1B receptor in Human [GtoPdb: 2] [UniProtKB: P28222]
  • This target only has 1 pki data point
  • 5.3
2 CHEMBL2027925_lig_chart_2 5-HT1B receptor Human
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  • 5-HT1D receptor in Human [GtoPdb: 3] [UniProtKB: P28221]
  • This target only has 1 pki data point
  • 5.1
3 CHEMBL2027925_lig_chart_3 5-HT1D receptor Human
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  • 5-HT2A receptor in Human [GtoPdb: 6] [UniProtKB: P28223]
  • This target only has 1 pki data point
  • 5.9
4 CHEMBL2027925_lig_chart_4 5-HT2A receptor Human
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  • 5-HT2B receptor in Human [GtoPdb: 7] [UniProtKB: P41595]
  • This target only has 1 pki data point
  • 5.8
5 CHEMBL2027925_lig_chart_5 5-HT2B receptor Human
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  • 5-HT2C receptor in Human [GtoPdb: 8] [UniProtKB: P28335]
  • This target only has 1 pki data point
  • 5.3
6 CHEMBL2027925_lig_chart_6 5-HT2C receptor Human
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  • 5-HT4 receptor in Human [GtoPdb: 9] [UniProtKB: Q13639]
  • This target only has 1 pki data point
  • 9.2
7 CHEMBL2027925_lig_chart_7 5-HT4 receptor Human
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  • 5-HT6 receptor in Human [GtoPdb: 11] [UniProtKB: P50406]
  • This target only has 1 pki data point
  • 5.6
8 CHEMBL2027925_lig_chart_8 5-HT6 receptor Human
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  • 5-HT7 receptor in Human [GtoPdb: 12] [UniProtKB: P34969]
  • This target only has 1 pki data point
  • 5.5
9 CHEMBL2027925_lig_chart_9 5-HT7 receptor Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
5-HT1A receptor in Human [GtoPdb: 1] [UniProtKB: P08908]
GtoPdb - - 6 pKi - - - J Pharmacol Exp Ther (2002) 302: 731-41 [PMID:12130738]
5-HT1B receptor in Human [GtoPdb: 2] [UniProtKB: P28222]
GtoPdb - - 5.3 pKi - - - J Pharmacol Exp Ther (2002) 302: 731-41 [PMID:12130738]
5-HT1D receptor in Human [GtoPdb: 3] [UniProtKB: P28221]
GtoPdb - - 5.1 pKi - - - J Pharmacol Exp Ther (2002) 302: 731-41 [PMID:12130738]
5-HT2A receptor in Human [GtoPdb: 6] [UniProtKB: P28223]
GtoPdb - - 5.9 pKi - - - J Pharmacol Exp Ther (2002) 302: 731-41 [PMID:12130738]
5-HT2B receptor in Human [GtoPdb: 7] [UniProtKB: P41595]
GtoPdb - - 5.8 pKi - - - J Pharmacol Exp Ther (2002) 302: 731-41 [PMID:12130738]
5-HT2C receptor in Human [GtoPdb: 8] [UniProtKB: P28335]
GtoPdb - - 5.3 pKi - - - J Pharmacol Exp Ther (2002) 302: 731-41 [PMID:12130738]
5-HT4 receptor in Human [GtoPdb: 9] [UniProtKB: Q13639]
GtoPdb - - 9.2 pKi - - - J Pharmacol Exp Ther (2002) 302: 731-41 [PMID:12130738]
5-HT6 receptor in Human [GtoPdb: 11] [UniProtKB: P50406]
GtoPdb - - 5.6 pKi - - - J Pharmacol Exp Ther (2002) 302: 731-41 [PMID:12130738]
5-HT7 receptor in Human [GtoPdb: 12] [UniProtKB: P34969]
GtoPdb - - 5.5 pKi - - - J Pharmacol Exp Ther (2002) 302: 731-41 [PMID:12130738]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]