zeltociclib [Ligand Id: 13754] activity data from GtoPdb

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  • cyclin dependent kinase 7 in Human [GtoPdb: 1979] [UniProtKB: P50613]
Created with Highcharts 10.3.3ValuesChart context menucyclin dependent kinase 7pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
cyclin dependent kinase 7 in Human [GtoPdb: 1979] [UniProtKB: P50613]
GtoPdb Inhibition of CDK7/CyclinH kinase activity - 7.7 pIC50 <20 nM IC50 WO2022134642A1. Aromatic heterocyclic compound, and pharmaceutical composition and application thereof (2022)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.