birelentinib [Ligand Id: 13735] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187] | ||||||||
| GtoPdb | Potency vs. BTKC481S | - | 9.07 | pIC50 | 0.86 | nM | IC50 | WO2021136219A1. Btk inhibitors (2021) |
| GtoPdb | Potency vs. WT hBTK | - | 9.15 | pIC50 | 0.7 | nM | IC50 | WO2021136219A1. Btk inhibitors (2021) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
