bosmolisib [Ligand Id: 13486] activity data from GtoPdb

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  • phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329]
Created with Highcharts 10.3.3ValuesChart context menuphosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit deltapKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736]
Created with Highcharts 10.3.3ValuesChart context menuphosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gammapKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329]
GtoPdb - - 8.7 pIC50 2 nM IC50 J Immunother Cancer (2022) 10: e003762 [PMID:35288465]
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736]
GtoPdb - - 7.82 pIC50 15 nM IC50 J Immunother Cancer (2022) 10: e003762 [PMID:35288465]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.