AMG487 [Ligand Id: 13071] activity data from GtoPdb

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  • CXCR3 in Human [GtoPdb: 70] [UniProtKB: P49682]
Created with Highcharts 10.3.3ValuesChart context menuCXCR3pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CXCR3 in Human [GtoPdb: 70] [UniProtKB: P49682]
GtoPdb Antagonism of 125I-IP10 binding to CXCR3 in a radioligand competition binding assay - 8.1 pIC50 8 nM IC50 Bioorg Med Chem Lett (2007) 17: 3339-43 [PMID:17448658]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.