pirotinib [Ligand Id: 12612] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| epidermal growth factor receptor in Human [GtoPdb: 1797] [UniProtKB: P00533] | ||||||||
| GtoPdb | - | - | 9 | pIC50 | 1 | nM | IC50 | WO2012027960A1. Quinazoline derivatives substituted by aniline, preparation method and use thereof (2012) |
| erb-b2 receptor tyrosine kinase 4 in Human [GtoPdb: 1799] [UniProtKB: Q15303] | ||||||||
| GtoPdb | - | - | 8.72 | pIC50 | 1.9 | nM | IC50 | WO2012027960A1. Quinazoline derivatives substituted by aniline, preparation method and use thereof (2012) |
| erb-b2 receptor tyrosine kinase 2 in Human [GtoPdb: 2019] [UniProtKB: P04626] | ||||||||
| GtoPdb | - | - | 8.19 | pIC50 | 6.5 | nM | IC50 | WO2012027960A1. Quinazoline derivatives substituted by aniline, preparation method and use thereof (2012) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
