compound 6li [Chan et al., 2022] [Ligand Id: 12249] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721] | ||||||||
| GtoPdb | - | - | 8.59 | pKd | 2.6 | nM | Kd | Journal of Nedicinal Chemistry (2022) : |
| fms related receptor tyrosine kinase 3 in Human [GtoPdb: 1807] [UniProtKB: P36888] | ||||||||
| GtoPdb | - | - | 8.6 | pKd | 2.5 | nM | Kd | Journal of Nedicinal Chemistry (2022) : |
| AXL receptor tyrosine kinase in Human [GtoPdb: 1835] [UniProtKB: P30530] | ||||||||
| GtoPdb | Binding affinity for hAXL | - | 9.59 | pKd | 0.26 | nM | Kd | Journal of Nedicinal Chemistry (2022) : |
| GtoPdb | Inhibition of kinase activity | - | 8.8 | pIC50 | 1.6 | nM | IC50 | Journal of Nedicinal Chemistry (2022) : |
| tyrosine kinase with immunoglobulin like and EGF like domains 1 in Human [GtoPdb: 1841] [UniProtKB: P35590] | ||||||||
| GtoPdb | - | - | 9.13 | pKd | 0.74 | nM | Kd | Journal of Nedicinal Chemistry (2022) : |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
