compound 11 [PMID: 35653642] [Ligand Id: 12047] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | Binding affinity for JAK2 JH1 (active kinase domain) | - | 5.47 | pKd | 3360 | nM | Kd | J Med Chem (2022) 65: 8380-8400 [PMID:35653642] |
| GtoPdb | Binding affinity for JAK2 JH2 wild-type | - | 7.12 | pKd | 75 | nM | Kd | J Med Chem (2022) 65: 8380-8400 [PMID:35653642] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
