tuxobertinib [Ligand Id: 11676] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| epidermal growth factor receptor in Human [GtoPdb: 1797] [UniProtKB: P00533] | ||||||||
| GtoPdb | Inhibition of WT EGFR kinase activity | - | 6.52 | pIC50 | 300 | nM | IC50 | US11034672B1. Tyrosine kinase inhibitor compositions, methods of making and methods of use (2021) |
| erb-b2 receptor tyrosine kinase 2 in Human [GtoPdb: 2019] [UniProtKB: P04626] | ||||||||
| GtoPdb | Inhibition of WT HER2 kinase activity | - | 8.3 | pIC50 | 5 | nM | IC50 | US11034672B1. Tyrosine kinase inhibitor compositions, methods of making and methods of use (2021) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
