edaxeterkib [Ligand Id: 11411] activity data from GtoPdb

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  • mitogen-activated protein kinase 1 in Human [GtoPdb: 1495] [UniProtKB: P28482]
  • This target only has 0 pki data point
  • 0
1 _lig_chart_1 mitogen-activated protein kinase 1 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
mitogen-activated protein kinase 1 in Human [GtoPdb: 1495] [UniProtKB: P28482]
GtoPdb Binned IC50 value from patent; determined using the proprietary Z'- LYTE kinase assay. - 7.3 pIC50 <50 nM IC50 WO2015051341A1. Inhibitors of erk and methods of use (2015)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.