CHMFL-PI4K-127 [Ligand Id: 11285] activity data from GtoPdb

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  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum [GtoPdb: 2972]
  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum 3D7 [GtoPdb: 2972] [UniProtKB: Q8I406]
  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum Dd2 [GtoPdb: 2972]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum [GtoPdb: 2972]
GtoPdb - - 9.05 pIC50 0.9 nM IC50 Eur J Med Chem (2020) 188: 112012 [PMID:31911293]
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum 3D7 [GtoPdb: 2972] [UniProtKB: Q8I406]
GtoPdb Parasite growth inhibition assay - 7.6 pEC50 25.1 nM EC50 Eur J Med Chem (2020) 188: 112012 [PMID:31911293]
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum Dd2 [GtoPdb: 2972]
GtoPdb Parasite growth inhibition assay - 7.52 pEC50 30.3 nM EC50 Eur J Med Chem (2020) 188: 112012 [PMID:31911293]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.