AZD3965 [Ligand Id: 10605] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Monocarboxylate transporter 1 in Human [GtoPdb: 988] [UniProtKB: P53985] | ||||||||
| GtoPdb | AZD3965 binding affinity to yeast membranes expressing recombinant human MCT1 by displacement of [3H]-MCT1 ligand. | - | 8.49 | pKi | 3.2 | nM | Ki | Oncotarget (2017) 8: 69219-69236 [PMID:29050199] |
| Monocarboxylate transporter 2 in Human [GtoPdb: 990] [UniProtKB: O60669] | ||||||||
| GtoPdb | AZD3965 binding affinity to yeast membranes expressing recombinant human MCT2 by displacement of [3H]-MCT2 ligand. | - | 7.7 | pKi | 20 | nM | Ki | Oncotarget (2017) 8: 69219-69236 [PMID:29050199] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
