carotegrast [Ligand Id: 10511] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| integrin α4β1 in Human [GtoPdb: 2580] | ||||||||
| GtoPdb | Measuring inhibition of binding between &alpha4;β1 integrin expressed by Jurkat cells and immobilised VCAM-1, in the presence of test compound. | - | 7.24 | pIC50 | 57 | nM | IC50 | US20110065918A1. New phenylalanine derivatives (2011) |
| integrin α4β7 in Human [GtoPdb: 2770] | ||||||||
| GtoPdb | Measuring inhibition of binding between &alpha4;β7 integrin expressed by RPMI-8866 cells and immobilised VCAM-1, in the presence of test compound. | - | 8.48 | pIC50 | 3.3 | nM | IC50 | US20110065918A1. New phenylalanine derivatives (2011) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
