AM-461 [Ligand Id: 10170] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| DP2 receptor in Human [GtoPdb: 339] [UniProtKB: Q9Y5Y4] | ||||||||
| GtoPdb | Radioligand ([3H]PGD2) displacement from human DP2 receptors expressed in HEK293 cells. | - | 8.28 | pIC50 | 5.2 | nM | IC50 | WO2011085033. DP2 ANTAGONIST AND USES THEREOF (2011) |
| DP2 receptor in Mouse [GtoPdb: 339] [UniProtKB: Q9Z2J6] | ||||||||
| GtoPdb | Radioligand ([3H]PGD2) displacement from mouse DP2 receptor. | - | 8.01 | pIC50 | 9.7 | nM | IC50 | WO2011085033. DP2 ANTAGONIST AND USES THEREOF (2011) |
| DP2 receptor in Rat [GtoPdb: 339] [UniProtKB: Q6XKD3] | ||||||||
| GtoPdb | Radioligand ([3H]PGD2) displacement from rat DP2 receptors. | - | 8.15 | pIC50 | 7 | nM | IC50 | WO2011085033. DP2 ANTAGONIST AND USES THEREOF (2011) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
