GSK963 [Ligand Id: 10132] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| receptor interacting serine/threonine kinase 1 in Human [GtoPdb: 2189] [UniProtKB: Q13546] | ||||||||
| GtoPdb | Inhibition of RIPK1 kinase activity in an ADP-Glo kinase assay measuring autophosphorylation of RIPK1 kinase domain in vitro; value calculated using a tight binding fit calculation. | - | 9.1 | pIC50 | 0.8 | nM | IC50 | Cell Death Discov (2015) 1: 15009 [PMID:27551444] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
