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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum V1/S [GtoPdb: 2972] | ||||||||
GtoPdb | Parasite growth inhibition assay | - | 8.38 | pIC50 | 4.2 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium berghei [GtoPdb: 2972] | ||||||||
GtoPdb | Parasite liver stage assay | - | 9.04 | pIC50 | 0.92 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium cynomolgi [GtoPdb: 2972] | ||||||||
GtoPdb | Parasite liver stage assay | - | 8 | pIC50 | <10 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum [GtoPdb: 2972] | ||||||||
GtoPdb | Parasite gametocyte viability assay | - | 6.87 | pIC50 | 134 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
GtoPdb | Standard membrane feeding assay (SMFA) | - | 7.02 | pIC50 | 96 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
GtoPdb | Parasite dual gamete formation assay (DGFA) | - | 7.1 | pIC50 | 80 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
GtoPdb | Parasite gametocyte viability assay | - | 7.18 | pIC50 | 66 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum K1 [GtoPdb: 2972] | ||||||||
GtoPdb | Parasite growth inhibition assay | - | 8.33 | pIC50 | 4.7 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum NF54 [GtoPdb: 2972] | ||||||||
GtoPdb | Parasite growth inhibition assay | - | 8.27 | pIC50 | 5.4 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum 7G8 [GtoPdb: 2972] | ||||||||
GtoPdb | Parasite growth inhibition assay | - | 8.39 | pIC50 | 4.1 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum Dd2 [GtoPdb: 2972] | ||||||||
GtoPdb | Parasite growth inhibition assay | - | 8.24 | pIC50 | 5.7 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum HB3 [GtoPdb: 2972] | ||||||||
GtoPdb | Parasite growth inhibition assay | - | 8.43 | pIC50 | 3.7 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum D6 [GtoPdb: 2972] | ||||||||
GtoPdb | Parasite growth inhibition assay | - | 8.28 | pIC50 | 5.2 | nM | IC50 | Antimicrob Agents Chemother (2018) 62: [PMID:29941635] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.