CM4620 [Ligand Id: 10087] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Orai1 in Human [GtoPdb: 2964] [UniProtKB: Q96D31] | ||||||||
| GtoPdb | In vitro inhibition of calcium entry mediated by Orai1/STIM1 CRAC channels. | - | 6.92 | pIC50 | 119 | nM | IC50 | WO2016138472A1. Pancreatitis treatment (2016) |
| Orai2 in Human [GtoPdb: 2965] [UniProtKB: Q96SN7] | ||||||||
| GtoPdb | In vitro inhibition of calcium entry mediated by Orai2/STIM1 CRAC channels. | - | 6.05 | pIC50 | 895 | nM | IC50 | WO2016138472A1. Pancreatitis treatment (2016) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
