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Benzodiazepine class drugs

Overview

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A list of approved drugs that modulate GABAA channel activity by binding to the allosteric benzodiazepine site. These drugs increase the inhibitory effects of GABA.

Ligands

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Ligands of relevance to immunopharmacology are highlighted in blue

alprazolam Show summary » More detailed page

chlordiazepoxide Show summary » More detailed page

clobazam Show summary » More detailed page

clonazepam Show summary » More detailed page

clorazepate Show summary » More detailed page

diazepam Show summary » More detailed page

estazolam Show summary » More detailed page

eszopiclone Show summary » More detailed page

flumazenil Show summary » More detailed page

flunitrazepam Show summary » More detailed page

flurazepam Show summary » More detailed page

halazepam Show summary » More detailed page

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lormetazepam Show summary » More detailed page

midazolam Show summary » More detailed page

oxazepam Show summary » More detailed page

quazepam Show summary » More detailed page

temazepam Show summary » More detailed page

triazolam Show summary » More detailed page

zaleplon Show summary » More detailed page

zolpidem Show summary » More detailed page

How to cite this family page

Database page citation:

Benzodiazepine class drugs. Accessed on 19/04/2024. IUPHAR/BPS Guide to PHARMACOLOGY, http://www.guidetopharmacology.org/GRAC/FamilyDisplayForward?familyId=1072.