|
|
|
D4 receptor
|
|
|
Hs |
Antagonist |
Antagonist |
9.3 |
pKi |
- |
3 |
|
⤷ |
pKi
9.3
[3]
|
α1B-adrenoceptor
|
|
|
Hs |
Antagonist |
Inverse agonist |
9.2 |
pKi |
- |
29 |
|
⤷ |
pKi
9.2
[29]
|
D3 receptor
|
|
|
Hs |
Antagonist |
Antagonist |
9.2 |
pKi |
- |
23 |
|
⤷ |
pKi
9.2
[23]
|
5-HT2A receptor
|
|
|
Rn |
Antagonist |
Antagonist |
9.0 – 9.2 |
pKi |
- |
4,21 |
|
⤷ |
pKi
9.0 – 9.2
[4,21]
|
D2 receptor
|
|
|
Rn |
Antagonist |
Antagonist |
8.4 – 9.4 |
pKi |
- |
12,14,23,25 |
|
⤷ |
pKi
8.4 – 9.4
[12,14,23,25]
|
5-HT2A receptor
|
|
|
Hs |
Antagonist |
Antagonist |
7.8 – 9.4 |
pKi |
- |
2,9,22 |
|
⤷ |
pKi
7.8 – 9.4
[2,9,22]
|
5-HT1B receptor
|
|
|
Mm |
Antagonist |
Antagonist |
8.3 |
pKi |
- |
13 |
|
⤷ |
pKi
8.3
[13]
|
α1A-adrenoceptor
|
|
|
Hs |
Antagonist |
Antagonist |
8.3 |
pKi |
- |
29 |
|
⤷ |
pKi
8.3
[29]
|
α1D-adrenoceptor
|
|
|
Hs |
Antagonist |
Antagonist |
8.1 |
pKi |
- |
29 |
|
⤷ |
pKi
8.1
[29]
|
5-HT7 receptor
|
|
|
Rn |
Antagonist |
Antagonist |
7.7 – 8.0 |
pKi |
- |
19-20 |
|
⤷ |
pKi
7.7 – 8.0
[19-20]
|
5-HT1A receptor
|
|
|
Hs |
Antagonist |
Antagonist |
6.7 – 8.8 |
pKi |
- |
15-17 |
|
⤷ |
pKi
6.7 – 8.8
[15-17]
|
5-HT7 receptor
|
|
|
Hs |
Antagonist |
Antagonist |
7.0 – 8.0 |
pKi |
- |
1,8,10 |
|
⤷ |
pKi
7.0 – 8.0
[1,8,10]
|
5-HT7 receptor
|
|
|
Mm |
Antagonist |
Antagonist |
7.2 |
pKi |
- |
18 |
|
⤷ |
pKi
7.2
[18]
|
D1 receptor
|
|
|
Hs |
Antagonist |
Antagonist |
6.7 |
pKi |
- |
24 |
|
⤷ |
pKi
6.7
[24]
|
5-HT2B receptor
|
|
|
Hs |
Antagonist |
Antagonist |
5.9 – 6.5 |
pKi |
- |
9,11,27 |
|
⤷ |
pKi
5.9 – 6.5
[9,11,27]
|
5-HT2C receptor
|
|
|
Hs |
Antagonist |
Antagonist |
5.6 – 6.2 |
pKi |
- |
5,7,9 |
|
⤷ |
pKi
5.6 – 6.2
[5,7,9]
|
5-HT6 receptor
|
|
|
Rn |
Antagonist |
Antagonist |
5.8 |
pKi |
- |
19 |
|
⤷ |
pKi
5.8
[19]
|
5-HT1D receptor
|
|
|
Hs |
Antagonist |
Antagonist |
5.5 – 6.0 |
pKi |
- |
6,28 |
|
⤷ |
pKi
5.5 – 6.0
[6,28]
|
5-HT2B receptor
|
|
|
Rn |
Antagonist |
Antagonist |
5.5 |
pKi |
- |
26 |
|
⤷ |
pKi
5.5
[26]
|
D5 receptor
|
|
|
Hs |
Antagonist |
Antagonist |
5.3 |
pKi |
- |
24 |
|
⤷ |
pKi
5.3
[24]
|
|