|
|
|
5-HT1A receptor
|
|
|
Hs |
Agonist |
Full agonist |
8.4 – 9.4 |
pKi |
- |
4,7,9,12,15,17-19 |
|
⤷ |
pKi
8.4 – 9.4
(Ki 3.98x10-9 – 3.98x10-10 M)
[4,7,9,12,15,17-19]
|
5-HT7 receptor
|
|
|
Rn |
Agonist |
Full agonist |
7.3 – 7.5 |
pKi |
- |
22-23 |
|
⤷ |
pKi
7.3 – 7.5
[22-23]
|
5-HT1D receptor
|
|
|
Hs |
Agonist |
Full agonist |
6.9 – 7.3 |
pKi |
- |
5,13,16 |
|
⤷ |
pKi
6.9 – 7.3
[5,13,16]
|
5-HT7 receptor
|
|
|
Hs |
Agonist |
Full agonist |
6.3 – 7.6 |
pKi |
- |
3,8,11,24 |
|
⤷ |
pKi
6.3 – 7.6
[3,8,11,24]
|
5-HT7 receptor
|
|
|
Mm |
Agonist |
Full agonist |
6.6 |
pKi |
- |
20 |
|
⤷ |
pKi
6.6
[20]
|
5-HT5A receptor
|
|
|
Mm |
Agonist |
Full agonist |
5.9 |
pKi |
- |
6,14 |
|
⤷ |
pKi
5.9
[6,14]
|
5-HT1F receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.8 |
pKi |
- |
1 |
|
⤷ |
pKi
5.8
[1]
|
5-HT5A receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.6 – 5.7 |
pKi |
- |
6,21 |
|
⤷ |
pKi
5.6 – 5.7
[6,21]
|
5-HT2A receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.6 |
pKi |
- |
10 |
|
⤷ |
pKi
5.6
[10]
|
5-HT2C receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.6 |
pKi |
- |
10 |
|
⤷ |
pKi
5.6
[10]
|
5-ht1e receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.5 |
pKi |
- |
1-2 |
|
⤷ |
pKi
5.5
[1-2]
|
5-HT2B receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.4 |
pKi |
- |
10 |
|
⤷ |
pKi
5.4
[10]
|
5-HT2B receptor
|
|
|
Rn |
Agonist |
Full agonist |
5.4 |
pKi |
- |
25 |
|
⤷ |
pKi
5.4
[25]
|
5-HT1B receptor
|
|
|
Hs |
Agonist |
Full agonist |
6.2 |
pIC50 |
- |
5 |
|
⤷ |
pIC50
6.2
[5]
|
|