Ligand id: 6892

Name: belatacept

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View more information in the IUPHAR Pharmacology Education Project: belatacept

View interactive charts of activity data from GtoPdb and ChEMBL (where available) across species

Bioactivity Comments
Belatacept binds to human CD86 with an IC50 of 0.102µg/mL and to CD80 with an IC50 of 0.009µg/mL [1].
Selectivity at other protein targets
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
CD80 Hs Inhibitor Inhibition - - - 1
Description: IC50= 0.009µg/mL
CD86 Hs Inhibitor Inhibition - - - 1
Description: IC50= 0.120µg/mL