R-715   Click here for help

GtoPdb Ligand ID: 661

Synonyms: [Ac-Lys-[d-βNal7,Ile8]des-Arg9]bradykinin | R 715 | R715
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
B1 receptor Hs Antagonist Antagonist 8.5 pA2 - 1
pA2 8.5 [1]
B1 receptor Hs Antagonist Antagonist 9.2 pKi - 2
pKi 9.2 (Ki 6.3x10-10 M) [2]
B1 receptor Mm Antagonist Antagonist 7.4 pKi - 2
pKi 7.4 [2]