tenalisib [Ligand Id: 9907] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336] | ||||||||
| GtoPdb | In a high throughput biochemical assay. | - | 5 | pIC50 | >10000 | nM | IC50 | US9790224B2. Dual selective PI3 delta and gamma kinase inhibitors (2017) |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta in Human [GtoPdb: 2154] [UniProtKB: P42338] | ||||||||
| GtoPdb | In a high throughput biochemical assay. | - | 5.4 | pIC50 | >4000 | nM | IC50 | US9790224B2. Dual selective PI3 delta and gamma kinase inhibitors (2017) |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329] | ||||||||
| GtoPdb | In a high throughput biochemical assay. | - | 7.62 | pIC50 | 24.05 | nM | IC50 | US9790224B2. Dual selective PI3 delta and gamma kinase inhibitors (2017) |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736] | ||||||||
| GtoPdb | In a high throughput biochemical assay. | - | 7.62 | pIC50 | 23.85 | nM | IC50 | US9790224B2. Dual selective PI3 delta and gamma kinase inhibitors (2017) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
