ChEMBL ligand: CHEMBL2064741
Peroxisome proliferator-activated receptor-γ/Peroxisome proliferator-activated receptor gamma in Human [ChEMBL: CHEMBL235] [GtoPdb: 595] [UniProtKB: P37231] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
Peroxisome proliferator-activated receptor-γ/Peroxisome proliferator-activated receptor gamma in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL235] [GtoPdb: 595] [UniProtKB: P37231]
ChEMBL	Agonist activity at PPARgamma LBD in human 293H DA cells after 16 hrs by TR-FRET activation reporter assay	F	6.33	pEC50	467	nM	EC50	J Med Chem (2012) 55: 4978-4989 [PMID:22582973]
ChEMBL	Binding affinity to PPARgamma LBD by fluorescence polarization based competitive binding assay	B	6.49	pEC50	325	nM	EC50	J Med Chem (2012) 55: 4978-4989 [PMID:22582973]
ChEMBL	Displacement of pan-PPAR fluormone from PPARgamma LBD by TR-FRET based LanthaScreen assay	B	6.67	pEC50	215	nM	EC50	J Med Chem (2012) 55: 4978-4989 [PMID:22582973]
GtoPdb	Measured by TR-FRET analysis.	-	6.67	pEC50	215	nM	EC50	J Med Chem (2012) 55: 4978-89 [PMID:22582973]

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]