α-NETA [Ligand Id: 9781] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1358898
  • chemerin receptor 1 in Human [GtoPdb: 79] [UniProtKB: Q99788]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
chemerin receptor 1 in Human [GtoPdb: 79] [UniProtKB: Q99788]
GtoPdb Antagonism of chemerin-stimulated β-arrestin 2 recruitment to CMKLR1 in a cellular assay. - 6.43 pIC50 375 nM IC50 PLoS ONE (2014) 9: e112925 [PMID:25437209]

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]