compound G1 [PMID: 36689364] [Ligand Id: 12354] activity data from GtoPdb

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  • epoxide hydrolase 2 in Human [GtoPdb: 2970] [UniProtKB: P34913]
  • epoxide hydrolase 2 in Mouse [GtoPdb: 2970] [UniProtKB: P34914]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
epoxide hydrolase 2 in Human [GtoPdb: 2970] [UniProtKB: P34913]
GtoPdb Inhibition of recombinant human sEH in vitro - 10.3 pIC50 0.05 nM IC50 J Med Chem (2023) 66: 2979-3009 [PMID:36689364]
epoxide hydrolase 2 in Mouse [GtoPdb: 2970] [UniProtKB: P34914]
GtoPdb Inhibition of recombinant mouse sEH in vitro - 9.85 pIC50 0.14 nM IC50 J Med Chem (2023) 66: 2979-3009 [PMID:36689364]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.