compound 14 [Schnute et al., 2023] [Ligand Id: 12351] activity data from GtoPdb

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  • RAR-related orphan receptor-γ in Human [GtoPdb: 600] [UniProtKB: P51449]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
RAR-related orphan receptor-γ in Human [GtoPdb: 600] [UniProtKB: P51449]
GtoPdb Inhibitory potency in a TR-FRET cofactor recruitment assay - 8.03 pIC50 9.3 nM IC50 ACS Medicinal Chemistry Letters (2023) :

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.