CXCR4 antagonist 22 [Ligand Id: 10146] activity data from GtoPdb

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  • CXCR4 in Human [GtoPdb: 71] [UniProtKB: P61073]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CXCR4 in Human [GtoPdb: 71] [UniProtKB: P61073]
GtoPdb Displacement of CXCR4-bound 125I-CXCL12 from membranes prepared from HEK293T cells expressing human CXCR4. - 6.3 pIC50 500 nM IC50 Eur J Med Chem (2019) 162: 631-649 [PMID:30476826]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.